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TQ0200 |
Paricalcitol
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Paricalcitol is a vitamin D receptor agonist. It is used for the prevention and treatment of secondary hyperparathyroidism associated with chronic renal failure. |
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T16015 |
Maxacalcitol
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22-Oxacalcitriol |
Others
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Maxacalcitol (22-Oxacalcitriol) is a ligand of VDR-like receptors and a non-serum calcium vitamin D3 analogue. Maxacalcitol inhibits parathyroid hormone (PTH) mRNA expression in vitro and in vivo. |
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T6430L |
Calcifediol monohydrate
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25-hydroxy Vitamin D3 monohydrate |
Endogenous Metabolite
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Calcifediol monohydrate (25-hydroxy Vitamin D3 monohydrate), the main circulating metabolite of vitamin D3, is a potent VDR inhibitor. |
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TQ0244 |
Calcipotriol monohydrate
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T14856 |
Calcipotriol
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MC 903,Calcipotriene |
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Calcipotriol (MC 903) is a synthetic VitD3 analogue. Which has a high affinity for the vitamin D receptor. |
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T6374 |
Alfacalcidol
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Bondiol,Etalpha,1-hydroxy Vitamin D3,1.alpha.-Hydroxyvitamin D3,1-hydroxycholecalciferol |
Others
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Alfacalcidol (Etalpha) (1-hydroxycholecalciferol; Alpha D3; 1.alpha.-Hydroxyvitamin D3) is a non-selective VDR activator medication. |
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T24166 |
Inecalcitol
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TX 522,TX-522,TX522 |
Apoptosis
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Inecalcitol (TX 522) is the growth inhibitor of human breast cancer cells. Inecalcitol is a unique vitamin D3 analog with Kd of 0.53 nM. |
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T6112 |
Doxercalciferol
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TSA 840,Hectorol,1.alpha.-Hydroxyvitamin D2,1α-hydroxyvitamin D2 |
Others
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Doxercalciferol (TSA 840) is a synthetic vitamin D2 analog, suppressing parathyroid synthesis and secretion, used to treat secondary hyperparathyroidism and metabolic bone disease. |
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T19559 |
Seocalcitol
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EB 1089 |
Others
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T19227 |
Calcitriol Impurities A
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Others
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Calcitriol Impurities A refers to the contaminants found in Calcitriol, the hormonally active metabolite of vitamin D3, which serves to activate the vitamin D receptor. |
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T11643 |
Impurity B of Calcitriol
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1β,25-Dihydroxyvitamin-D3,1-Epicalcitriol |
Others
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Impurity B of Calcitriol is an impurity of Calcitriol. Calcitriol is the hormonally active form of vitamin D, Calcitriol is the active metabolite of vitamin D3 that activates the vitamin D receptor (VDR). |
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T23762 |
Atocalcitol
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Atocalcitol is a vitamin D analog. It also acts as an agonist of alcitriol receptor. |
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T10663 |
Calcitriol-d6
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Calcitriol D6 |
Others
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Calcitriol D6 is the deuterated form of Calcitriol, which is the hormonally active form of vitamin D. Calcitriol is the active metabolite of vitamin D3 that activates the vitamin D receptor. |
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T13197 |
Trans-Doxercalciferol
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Others
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trans-Doxercalciferol is an isomer of Doxercalciferol. Doxercalciferol is an activator of the Vitamin D receptor and prevents renal disease. |
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T27825 |
LG190178
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LG-190178,LG 190178 |
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LG190178, a vitamin D receptor (VDR) ligand, is a therapeutic agent used for the treatment of psoriasis, osteoporosis, and secondary hyperparathyroidism. |
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T11089 |
Doxercalciferol-D3
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Others
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Doxercalciferol-d3 is the deuterated form of Doxercalciferol and ACTS as vitamin D receptor activator (VDRA), which is a vitamin D2 analogue. |
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T78944 |
VDR agonist 2
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VDR agonist 2 (compound 16i), a vitamin D receptor (VDR) agonist, effectively inhibits TGF-β1-induced hepatic stellate cell (HSC) activation, demonstrating notable anti-hepatic fibrosis efficacy both in vitro and in vivo... |
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T69676 |
LG190155
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LG190155 is a moderately potent VDR agonist. Vitamin D receptor (VDR) agonists are well known for their capacity to control calcium and bone metabolism and to regulate growth and differentiation of many cell types. |
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T35524 |
(1S)-Calcitriol
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(1S)-Calcitriol (1α,25-Dihydroxy-3-epi-vitamin-D3), a natural metabolite of 1α,25-dihydroxyvitamin D3 (1α,25(OH)2D3), exerts potent actions through vitamin D receptor (VDR) activation, including the inhibition of keratin... |
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T24407 |
LG190119
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LG-190119,LG 190119 |
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LG190119 is a nonsecosteroidal vitamin D receptor modulator. It effectively inhibited LNCaP xenograft tumor growth without increased serum calcium levels or any other apparent side effects. It also inhibits the growth of... |
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T36593 |
TEI-9648
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TEI-9648, an analogue of Vitamin D3 Lactone, acts as a potent and specific antagonist to the vitamin D receptor (VDR). This compound effectively blocks the genomic actions mediated by VDR and the Vitamin D responsive ele... |
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T13292 |
VDR agonist 1
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Others
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VDR agonist 1 (compound 28), a nonsteroidal Vitamin D receptor (VDR) agonist, demonstrates potent activity with a low IC 50 of 690 nM in MCF-7 cells. It inhibits cell cycle progression through upregulation of p21 and p27... |
